Structural studies of 4-aminoantipyrine derivatives

Detalhes bibliográficos
Autor(a) principal: Cunha, Silvio do Desterro
Data de Publicação: 2005
Outros Autores: Oliveira, Shana M., Rodrigues Jr, Manoel T., Bastos, Rodrigo M., Ferrari, Jailton, Oliveira, Cecília M.A. de, Kato, Lucília, Napolitano, Hamilton B., Vencato, Ivo, Lariucci, Carlito
Tipo de documento: Artigo
Idioma: eng
Título da fonte: Repositório Institucional da UFBA
Texto Completo: http://repositorio.ufba.br/ri/handle/ri/13542
Resumo: Texto completo: acesso restrito. p.32–39
id UFBA-2_e9e0f9948cf48db5c4d24bc1517c45af
oai_identifier_str oai:repositorio.ufba.br:ri/13542
network_acronym_str UFBA-2
network_name_str Repositório Institucional da UFBA
repository_id_str 1932
spelling Cunha, Silvio do DesterroOliveira, Shana M.Rodrigues Jr, Manoel T.Bastos, Rodrigo M.Ferrari, JailtonOliveira, Cecília M.A. deKato, LucíliaNapolitano, Hamilton B.Vencato, IvoLariucci, CarlitoCunha, Silvio do DesterroOliveira, Shana M.Rodrigues Jr, Manoel T.Bastos, Rodrigo M.Ferrari, JailtonOliveira, Cecília M.A. deKato, LucíliaNapolitano, Hamilton B.Vencato, IvoLariucci, Carlito2013-11-04T11:43:29Z20050022-2860http://repositorio.ufba.br/ri/handle/ri/13542v.752 n. 1-3Texto completo: acesso restrito. p.32–39Reaction of 4-aminoantipyrine with acetylacetone, ethyl acetoacetate, benzoyl isothiocyanate, phenyl isothiocyanate, maleic anhydride and methoxymethylene Meldrum's acid afforded a series of new antipyrine derivatives. The antibacterial activity of the synthesized compounds against Micrococcus luteus ATCC 9341, Staphilococcus aureus ATCC 29737, and Escherichia coli ATCC 8739 was evaluated and the minimal inhibitory concentration determined. Modest activity was found only to the maleamic acid obtained from the reaction of 4-aminoantipyrine and maleic anhydride. 1H NMR investigation of this maleamic acid showed that it is slowly converted to the corresponding toxic maleimide. The structures of three derivatives were determined by X-ray diffraction analysis.Submitted by Edileide Reis (leyde-landy@hotmail.com) on 2013-11-04T11:43:29Z No. of bitstreams: 1 Silvio Cunha.pdf: 266922 bytes, checksum: 4445b82708b0cf11f9e50dce2fab1938 (MD5)Made available in DSpace on 2013-11-04T11:43:29Z (GMT). No. of bitstreams: 1 Silvio Cunha.pdf: 266922 bytes, checksum: 4445b82708b0cf11f9e50dce2fab1938 (MD5) Previous issue date: 2005http://dx.doi.org.ez10.periodicos.capes.gov.br/10.1016/j.molstruc.2005.05.016reponame:Repositório Institucional da UFBAinstname:Universidade Federal da Bahia (UFBA)instacron:UFBAEnaminonesThioureasMeleimideStructural studies of 4-aminoantipyrine derivativesJournal of Molecular Structureinfo:eu-repo/semantics/publishedVersioninfo:eu-repo/semantics/article10000-01-01info:eu-repo/semantics/openAccessengORIGINALSilvio Cunha.pdfSilvio Cunha.pdfapplication/pdf266922https://repositorio.ufba.br/bitstream/ri/13542/1/Silvio%20Cunha.pdf4445b82708b0cf11f9e50dce2fab1938MD51LICENSElicense.txtlicense.txttext/plain1383https://repositorio.ufba.br/bitstream/ri/13542/2/license.txt05eca2f01d0b3307819d0369dab18a34MD52TEXTSilvio Cunha.pdf.txtSilvio Cunha.pdf.txtExtracted texttext/plain24917https://repositorio.ufba.br/bitstream/ri/13542/3/Silvio%20Cunha.pdf.txtf4ff994ff1156c87e69fe62433f9c408MD53ri/135422022-08-08 13:17:50.0oai:repositorio.ufba.br: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ório InstitucionalPUBhttp://192.188.11.11:8080/oai/requestopendoar:19322022-08-08T16:17:50Repositório Institucional da UFBA - Universidade Federal da Bahia (UFBA)false
dc.title.pt_BR.fl_str_mv Structural studies of 4-aminoantipyrine derivatives
dc.title.alternative.pt_BR.fl_str_mv Journal of Molecular Structure
title Structural studies of 4-aminoantipyrine derivatives
spellingShingle Structural studies of 4-aminoantipyrine derivatives
Cunha, Silvio do Desterro
Enaminones
Thioureas
Meleimide
title_short Structural studies of 4-aminoantipyrine derivatives
title_full Structural studies of 4-aminoantipyrine derivatives
title_fullStr Structural studies of 4-aminoantipyrine derivatives
title_full_unstemmed Structural studies of 4-aminoantipyrine derivatives
title_sort Structural studies of 4-aminoantipyrine derivatives
author Cunha, Silvio do Desterro
author_facet Cunha, Silvio do Desterro
Oliveira, Shana M.
Rodrigues Jr, Manoel T.
Bastos, Rodrigo M.
Ferrari, Jailton
Oliveira, Cecília M.A. de
Kato, Lucília
Napolitano, Hamilton B.
Vencato, Ivo
Lariucci, Carlito
author_role author
author2 Oliveira, Shana M.
Rodrigues Jr, Manoel T.
Bastos, Rodrigo M.
Ferrari, Jailton
Oliveira, Cecília M.A. de
Kato, Lucília
Napolitano, Hamilton B.
Vencato, Ivo
Lariucci, Carlito
author2_role author
author
author
author
author
author
author
author
author
dc.contributor.author.fl_str_mv Cunha, Silvio do Desterro
Oliveira, Shana M.
Rodrigues Jr, Manoel T.
Bastos, Rodrigo M.
Ferrari, Jailton
Oliveira, Cecília M.A. de
Kato, Lucília
Napolitano, Hamilton B.
Vencato, Ivo
Lariucci, Carlito
Cunha, Silvio do Desterro
Oliveira, Shana M.
Rodrigues Jr, Manoel T.
Bastos, Rodrigo M.
Ferrari, Jailton
Oliveira, Cecília M.A. de
Kato, Lucília
Napolitano, Hamilton B.
Vencato, Ivo
Lariucci, Carlito
dc.subject.por.fl_str_mv Enaminones
Thioureas
Meleimide
topic Enaminones
Thioureas
Meleimide
description Texto completo: acesso restrito. p.32–39
publishDate 2005
dc.date.issued.fl_str_mv 2005
dc.date.accessioned.fl_str_mv 2013-11-04T11:43:29Z
dc.type.status.fl_str_mv info:eu-repo/semantics/publishedVersion
dc.type.driver.fl_str_mv info:eu-repo/semantics/article
format article
status_str publishedVersion
dc.identifier.uri.fl_str_mv http://repositorio.ufba.br/ri/handle/ri/13542
dc.identifier.issn.none.fl_str_mv 0022-2860
dc.identifier.number.pt_BR.fl_str_mv v.752 n. 1-3
identifier_str_mv 0022-2860
v.752 n. 1-3
url http://repositorio.ufba.br/ri/handle/ri/13542
dc.language.iso.fl_str_mv eng
language eng
dc.rights.driver.fl_str_mv info:eu-repo/semantics/openAccess
eu_rights_str_mv openAccess
dc.source.pt_BR.fl_str_mv http://dx.doi.org.ez10.periodicos.capes.gov.br/10.1016/j.molstruc.2005.05.016
dc.source.none.fl_str_mv reponame:Repositório Institucional da UFBA
instname:Universidade Federal da Bahia (UFBA)
instacron:UFBA
instname_str Universidade Federal da Bahia (UFBA)
instacron_str UFBA
institution UFBA
reponame_str Repositório Institucional da UFBA
collection Repositório Institucional da UFBA
bitstream.url.fl_str_mv https://repositorio.ufba.br/bitstream/ri/13542/1/Silvio%20Cunha.pdf
https://repositorio.ufba.br/bitstream/ri/13542/2/license.txt
https://repositorio.ufba.br/bitstream/ri/13542/3/Silvio%20Cunha.pdf.txt
bitstream.checksum.fl_str_mv 4445b82708b0cf11f9e50dce2fab1938
05eca2f01d0b3307819d0369dab18a34
f4ff994ff1156c87e69fe62433f9c408
bitstream.checksumAlgorithm.fl_str_mv MD5
MD5
MD5
repository.name.fl_str_mv Repositório Institucional da UFBA - Universidade Federal da Bahia (UFBA)
repository.mail.fl_str_mv
_version_ 1798057643025104896